Journal of Medicinal Chemistry
Volume 41, Issue 4 (February 12, 1998)
Copyright © 1998
American Chemical Society
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407-412 | Identification and Initial Structure-Activity Relationships of (R)-5-(2-Azetidinylmethoxy)-2-chloropyridine (ABT-594), a Potent, Orally Active, Non-Opiate Analgesic Agent Acting via Neuronal Nicotinic Acetylcholine Receptors
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413-419 | 2-Chloro-4-(trifluoromethyl)pyrimidine-5-N-(3',5'-bis(trifluoromethyl)phenyl)- carboxamide: A Potent Inhibitor of NF- B- and AP-1-Mediated Gene Expression Identified Using Solution-Phase Combinatorial Chemistry
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ARTICLES | |
420-427 | Design, Synthesis, and Biological Evaluation of Conformationally Constrained aci-Reductone Mimics of Arachidonic Acid
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428-436 | Specificity of Diastereomers of [99mTc]TRODAT-1 as Dopamine Transporter Imaging Agents
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437-450 | Identification and Initial Structure-Activity Relationships of a Novel Class of Nonpeptide Inhibitors of Blood Coagulation Factor Xa
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451-467 | Mapping the Melatonin Receptor. 5. Melatonin Agonists and Antagonists Derived from Tetrahydrocyclopent[b]indoles, Tetrahydrocarbazoles and Hexahydrocyclohept[b]indoles
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468-477 | Rigid Phencyclidine Analogues. Binding to the Phencyclidine and  1 Receptors
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478-488 | Random or Rational Design? Evaluation of Diverse Compound Subsets from Chemical Structure Databases
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489-502 | Novel Non-Peptide Fibrinogen Receptor Antagonists. 1. Synthesis and Glycoprotein IIb-IIIa Antagonistic Activities of 1,3,4-Trisubstituted 2-Oxopiperazine Derivatives Incorporating Side-Chain Functions of the RGDF Peptide
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503-508 | Inhibition of Human O6-Alkylguanine-DNA Alkyltransferase and Potentiation of the Cytotoxicity of Chloroethylnitrosourea by 4(6)-(Benzyloxy)-2,6(4)-diamino-5-(nitro or nitroso)pyrimidine Derivatives and Analogues
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509-514 | Synthesis and Calcium Channel-Modulating Effects of Alkyl (or Cycloalkyl) 1,4-Dihydro-2,6-dimethyl-3-nitro-4-pyridyl-5-pyridinecarboxylate Racemates and Enantiomers
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515-529 | The Partitioning of Phosphoramide Mustard and Its Aziridinium Ions among Alkylation and P-N Bond Hydrolysis Reactions
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530-539 | N-{trans-2-[[2'-(Acetylamino)cyclohexyl]oxy]acetyl}-L-alanyl-D-glutamic Acid: A Novel Immunologically Active Carbocyclic Muramyl Dipeptide Analogue
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540-554 | 29-Methylidene-2,3-oxidosqualene Derivatives as Stereospecific Mechanism-Based Inhibitors of Liver and Yeast Oxidosqualene Cyclase
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555-563 | A1 Adenosine Receptor Antagonists as Ligands for Positron Emission Tomography (PET) and Single-Photon Emission Tomography (SPET)
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564-578 | A Novel Class of Orally Active Non-Peptide Bradykinin B2 Receptor Antagonists. 1. Construction of the Basic Framework
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579-590 | Synthesis and Anticonvulsant Activity of a New Class of 2-[(Arylalkyl)amino]alkanamide Derivatives
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591-601 | Asymmetric Synthesis and Pharmacology of Methylphenidate and Its Para-Substituted Derivatives
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602-617 | Discovery of Ritonavir, a Potent Inhibitor of HIV Protease with High Oral Bioavailability and Clinical Efficacy
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618-622 | Synthesis of a Methylenebis(phosphonate) Analogue of Mycophenolic Adenine Dinucleotide: A Glucuronidation-Resistant MAD Analogue of NAD
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623-639 | Synthesis and Biological Activity of a Novel Series of Nonsteroidal, Peripherally Selective Androgen Receptor Antagonists Derived from 1,2-Dihydropyridono[5,6-g]quinolines
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640-649 | Highly Selective and Orally Active Inhibitors of Type IV Collagenase (MMP-9 and MMP-2): N-Sulfonylamino Acid Derivatives
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NOTES | |
650-652 | Effects of  - and  -Galactosylated C2-Ceramides on the Immune System
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BOOK REVIEWS | |
653-653 | Recent Developments in Theoretical Studies of Proteins Edited by Ron Elber. World Scientific Publishing Co. Pte. Ltd., Singapore. 1996. viii + 399 pp. 16 × 22 cm. ISBN 981-02-2196-7. $78.00.
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653-654 | ACCORD Synopsys Scientific Systems Ltd., United Kingdom. Version 2.0 for Windows.  495 (295 academic price).
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654-654 | HPLC Methods for Pharmaceutical Analysis By George Lunn and Norman R. Schmuff. John Wiley and Sons, Inc., New York. 1997. xxii + 1609 pp. 19 × 26 cm. ISBN 0-471-18176-5. $150.00.
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